Arid
DOI10.1080/14786419.2013.856904
Brazilian brown propolis elicits antileishmanial effect against promastigote and amastigote forms of Leishmania amazonensis
Santana, Lorena C. L. R.1; Carneiro, Sabrina Maria P.1; Caland-Neto, Laurentino B.2; Arcanjo, Daniel D. R.1; Moita-Neto, Jose M.2; Cito, Antonia M. G. L.2; Carvalho, Fernando Aecio A.1,3
通讯作者Carvalho, Fernando Aecio A.
来源期刊NATURAL PRODUCT RESEARCH
ISSN1478-6419
EISSN1478-6427
出版年2014
卷号28期号:5页码:340-343
英文摘要

Propolis is a complex matrix of chemical constituents extracted from plants and produced by bees which is used in folk medicine due to its several pharmacological properties. Its chemical composition varies according to the region where it is produced. This work has studied the antileishmanial activity and cytotoxicity of brown propolis (BP) originating from the semi-arid region of Piaui, Brazil. The BP showed significant inhibition of the Leishmania amazonensis promastigotes growth as well as being effective in reducing infection of murine macrophages and the number of internalised amastigotes in these cells. The dichloromethane fraction was the most active and showed the best selectivity index. The studied samples presented good activity and the fractioning improved the antileishmanial activity without an increase in the cytotoxicity against mammalian cells. Therefore, BP is a potential source for development of apitherapeutic products for the treatment of leishmaniasis.


英文关键词leishmaniasis antiparasitic activity cytotoxicity propolis brown propolis
类型Article
语种英语
国家Brazil
收录类别SCI-E
WOS记录号WOS:000333994100012
WOS类目Chemistry, Applied ; Chemistry, Medicinal
WOS研究方向Chemistry ; Pharmacology & Pharmacy
资源类型期刊论文
条目标识符http://119.78.100.177/qdio/handle/2XILL650/183948
作者单位1.Univ Fed Piaui, Med Plants Res Ctr, Teresina, PI, Brazil;
2.Univ Fed Piaui, Dept Chem, Teresina, PI, Brazil;
3.Univ Fed Piaui, Dept Biochem & Pharmacol, Teresina, PI, Brazil
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GB/T 7714
Santana, Lorena C. L. R.,Carneiro, Sabrina Maria P.,Caland-Neto, Laurentino B.,et al. Brazilian brown propolis elicits antileishmanial effect against promastigote and amastigote forms of Leishmania amazonensis[J],2014,28(5):340-343.
APA Santana, Lorena C. L. R..,Carneiro, Sabrina Maria P..,Caland-Neto, Laurentino B..,Arcanjo, Daniel D. R..,Moita-Neto, Jose M..,...&Carvalho, Fernando Aecio A..(2014).Brazilian brown propolis elicits antileishmanial effect against promastigote and amastigote forms of Leishmania amazonensis.NATURAL PRODUCT RESEARCH,28(5),340-343.
MLA Santana, Lorena C. L. R.,et al."Brazilian brown propolis elicits antileishmanial effect against promastigote and amastigote forms of Leishmania amazonensis".NATURAL PRODUCT RESEARCH 28.5(2014):340-343.
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