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Reconciling the lock-and-key and dynamic views of canonical serine protease inhibitor action 期刊论文
发表期刊: FEBS LETTERS. 出版年: 2010, 卷号: 584, 期号: 1, 页码: 203-206
作者:  Gaspari, Zoltan;  Varnai, Peter;  Szappanos, Balazs;  Perczel, Andras
收藏  |  浏览/下载:17/0  |  提交时间:2019/11/29
Canonical serine protease inhibitor  Nanosecond-timescale conformer selection  Protease binding  Internal dynamics  Dynamic conformational ensemble  Population shift  
Extended intermolecular interactions in a serine protease-canonical inhibitor complex account for strong and highly specific inhibition 期刊论文
发表期刊: JOURNAL OF MOLECULAR BIOLOGY. 出版年: 2005, 卷号: 350, 期号: 1, 页码: 156-169
作者:  Fodor, K;  Harmat, V;  Hetenyi, C;  Kardos, J;  Antal, J;  Perczel, A;  Patthy, A;  Katona, G;  Graf, L
收藏  |  浏览/下载:12/0  |  提交时间:2019/11/28
serine protease  canonical inhibitor  X-ray crystallography  NMR  specificity